제품 요약
Antide (CAS 112568-12-4) Product Details Antide, with CAS Number 112568-12-4, is a potent synthetic GnRH (Gonadotropin-Releasing Hormone) antagonist, also known as Antide Acetate. It is a linear modified peptide with N-terminal acetylation and C-terminal amidation, which significantly enhances its ...
GMP factory supply high purity Antide peptide CAS 112568-12-4 Antide powder for research
기본 특성
원산지:
무한
브랜드 이름:
Bovita
인증:
DMF
모델 번호:
BVR14
부동산 거래
최소 주문 수량:
1G
가격:
220USD
표준 포장:
PVC 병 또는 알루미늄 호일 백
배달 시간:
3~7일
지불 조건:
L/C,D/A,D/P,T/T,웨스턴 유니온
공급 능력:
5kg/월
제품 상세정보
강조하다:
GMP Antide peptide powder
,high purity Antide peptide
,research Antide peptide powder
Appearence:
가루
Specification:
1g/5g/가방
Stocks:
예
Storage Temp:
2~8°C
Test Method:
HPLC HNMR
Color:
하얀색
Casnumber:
펩타이드에 따라 다름
Puritylevel:
제약 등급
Einecs:
112568-12-4
Lead Time:
지불 후 3-5 일
Product Type:
맞춤형 펩타이드
Packagingmaterial:
PVC 병 또는 알루미늄 호일 백
Type:
GLP-2
제품 설명
세부 사양 및 특징
Antide (CAS 112568-12-4) Product Details
Antide, with CAS Number 112568-12-4, is a potent synthetic GnRH (Gonadotropin-Releasing Hormone) antagonist, also known as Antide Acetate. It is a linear modified peptide with N-terminal acetylation and C-terminal amidation, which significantly enhances its stability and biological activity. As a high-purity peptide hormone, it strictly complies with international pharmaceutical standards (GMP, USP, EP) and is widely used in global medical research, clinical trials and pharmaceutical R&D, especially in the fields of hormone-related disease treatment and reproductive medicine research.
Product Basic Information
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Item
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Details
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CAS Number
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112568-12-4
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Product Name
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Antide; Antide Acetate; GnRH Antagonist
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Chemical Formula
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C₈₂H₁₀₈ClN₁₇O₁₄
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Molecular Weight
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Approx. 1591.29
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Appearance
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White to Off-White Solid Powder
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Purity
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≥98% (HPLC); ≥99% available for research grade
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Solubility
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Approx. 10 mg/mL in Water (ultrasonic assistance recommended); Soluble in appropriate organic solvents
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Storage Condition
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Sealed, Protected from Light; -80°C for 2 years, -20°C for 1 year (powder); -80°C for 6 months, -20°C for 1 month (dissolved); Avoid repeated freeze-thaw cycles
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Shelf Life
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24 Months under Proper Storage Conditions (powder)
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Peptide Sequence
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Ac-D-2Nal-pCl-D-Phe-D-3Pal-S-K(nic)-D-K(nic)-L-K(iPr)-P-D-Ala-NH₂
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Pharmacological Action & Clinical Applications
Mechanism of Action
Antide acts as a potent GnRH antagonist by competitively binding to GnRH receptors in the anterior pituitary gland, blocking the binding of endogenous GnRH to its receptors. This binding inhibits the release of luteinizing hormone (LH) and follicle-stimulating hormone (FSH), thereby reducing the synthesis and secretion of gonadal hormones. In males, it can lower levels to castration-like levels, while in females, it affects the secretion of and progesterone. Its long-acting effect is attributed to its binding to serum proteins, which slows its clearance in the circulatory system, with a half-life of approximately 6.5 days in the second phase after intravenous injection.
Main Clinical Uses
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Oncology Research: Potential application in the treatment of -dependent diseases such as prostate cancer, by reducing levels through inhibiting LH and FSH release.
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Reproductive Medicine Research: Used to study the regulation of the reproductive endocrine axis, and as a research tool for developing new GnRH antagonist drugs, similar to Cetrorelix and Ganirelix but with distinct pharmacokinetic properties.
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Animal Model Research: Widely used in animal experiments (such as male rats and cynomolgus monkeys) to induce long-term inhibition of gonadal function, with dose-dependent effects on LH, levels and reproductive organ weight.
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Pharmaceutical R&D: Serves as a key tool for researching the GnRH receptor pathway and developing new drugs for hormone-related diseases.
Contraindications & Adverse Reactions
Contraindications: Prohibited for patients with hypersensitivity to any component of the product, pregnant or lactating women, and those with severe hepatic or renal impairment.
Adverse Reactions: Common reactions may include transient hormonal disorders, hot flashes, fatigue and mild gastrointestinal discomfort. Long-term use may lead to gonadal function inhibition and related complications. Regular monitoring of hormone levels, hepatic and renal function is recommended during use.
Export Compliance & Trade Information
Regulatory Attribute
Antide is classified as a peptide hormone drug in China, subject to the administration of Drug Import and Export License (Regulatory Code: L). It complies with GMP, USP, EP and other international pharmaceutical standards, and meets the regulatory requirements of major global markets such as the EU and the United States, including Export Administration Regulations (EAR) for the US market.
HS Code & Declaration Elements
Recommended HS Code: 2937190090 (Other peptide hormones; subject to the latest customs code of the importing country); For finished dosage forms, refer to HS Code 3004 (Medicaments for therapeutic or prophylactic uses). Note that ECCN (Export Control Classification Number) is distinct from HS Code and should be confirmed based on local regulations for US exports.
Declaration Elements: CAS Number, Product Name, Purity, Usage (Medical/Research), Composition, Brand, Peptide Sequence, Modification Information (N-terminal acetylation, C-terminal amidation), etc.
Export Documentation Requirements
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Drug Export Sales Certificate (valid for 3 years), issued by the provincial drug regulatory authority of China.
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Import License or official certification of the importing country (if required), especially complying with FDA regulations for the US market, CEP requirements for the EU market, and EAR requirements for US exports.
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Relevant qualifications: GMP Certificate, Production Approval Number, Sales Contract, etc.
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Test Reports: COA (Certificate of Analysis), MSDS (Material Safety Data Sheet), peptide sequence verification report, purity test report (HPLC/MS).
Logistics & Packaging
Packaging: Aluminum foil bag or glass vial, labeled with "Drug, Do Not Freeze, Protect from Light", peptide sequence and modification information; sealed packaging to prevent moisture, contamination and peptide degradation.
Transportation: Cold chain transportation is recommended (shipping with blue ice) to ensure the product quality during transportation; the whole process is temperature-controlled and traceable; avoid extreme temperature changes and repeated freeze-thaw cycles. Ambient temperature shipping is acceptable for short-distance transportation with proper packaging.
Quality Assurance & After-Sales Service
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Strict Quality Control: Each batch of products undergoes HPLC, MS and peptide sequence verification tests to ensure purity, stability and structural accuracy; endotoxin testing is available upon request.
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Customized Service: We can provide customized packaging and specifications according to customer needs, including small-volume research-grade products (≥99% purity) and large-volume medical-grade products.
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After-Sales Support: Provide professional technical guidance (including reconstitution and storage instructions), timely solve logistics and customs clearance problems, and ensure smooth trade; provide relevant regulatory compliance guidance for specific markets (such as ECCN confirmation for US exports).
Note
For Medical/Research Use Only. Not for use as health supplements or for illegal purposes. Customers must have legal drug import qualifications in their country/region and comply with local regulatory requirements (such as FDA regulations, EU laws and EAR for US exports). We will not be liable for any risks caused by non-compliant use or import.
If you need more detailed technical data, customized specifications or export compliance guidance for specific countries (such as EU, USA), please contact us directly.

전체 평점
스타 5명
100%
별 4개
0
3 별
0
별 2개
0
별 1개
0
모든 리뷰
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Jvery good high purity, good use
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Jquick shipment, thanks
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Agood quality, safety shipment
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